Synthesis and activity of 3-epi-actinobolin.
نویسندگان
چکیده
3-epi-Actinobolin was synthesized by the chemical transformation of actinobolin involving a key step of the reconstruction of fused delta-lacton skeleton via intramolecular acylation reaction. The analogue with low toxicity weakly inhibits Gram-positive and Gram-negative bacteria.
منابع مشابه
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ورودعنوان ژورنال:
- The Journal of antibiotics
دوره 51 2 شماره
صفحات -
تاریخ انتشار 1998